Compound 1
|
− 6.4
|
Glu-50
|
Pro-79
|
Asp-73, Asn-46, Ala-47, Arg-76, Gly-77, Ile-78, Gly-81, Ile-94, Arg-136, Thr-165
|
Compound 2
|
− 6.7
|
Gly-77, Thr-165
|
Glu-50
|
Asp-73, Ile-78, Ile-94
|
Compound 3
|
− 6.9
|
Gly-77, Asn-46, Thr-165
|
–
|
Asp-73, Ala-47, Asp-49, Glu-50, Gly-75, Arg-76, Ile-78, Pro-79, Ile-94, Arg-136
|
Compound 4
|
− 5.6
|
Asp-73
|
Ile-78
|
Asn-46, Ala-47, Glu-50, Arg-76, Gly-77, Pro-79, Ile-94, Thr-165
|
Compound 5
|
− 6.5
|
Asp-73
|
Ile-78, Pro-79, Ile-94
|
Asn-46, Ala-47, Glu-50, Arg-76, Gly-77, Arg-136, Thr-165,
|
Ciprofloxacin
|
− 6.9
|
Asp-73, Asn-46, Arg-76
|
Ile-78, Ile-94, Glu-50, Gly-77
|
Ala-47, Pro-79, Thr-165
|