From: Pharmacological significance of heterocyclic 1H-benzimidazole scaffolds: a review
Comp. | IβHS | IC50 (µM) | IGP | % P | SD |
---|---|---|---|---|---|
30a | 95.43 ± 0.58 | 8.43 | 0 | 4.02 ± 0.45 | 17 ± 1.26 |
30b | 75.76 ± 0.99 | 11.10 | 14.08 ± 0.88 | 1.8 ± 0.49 | 18.8 ± 2.05 |
Leupeptin | – | – | 91.62 ± 0.69 | – | – |
Pepstatin | – | – | 95.45 ± 0.66 | – | – |
Chloroquine | 94.19 ± 0.36 | – | 24.12 ± 1.16 | 1.3 ± 0.3 | > 30 |
Saline Solution | – | – | – | 21.8 ± 2.31 | 11.66 ± 1.66 |