5
|
− 11.054
|
− 68.766
|
Gln455, Ser452, Ala451, Val448, Val445, Asn383, Tyr386, Hie387, Trp388, Hie389, Leu391, Leu392, Phe396, Phe405, Val296, Leu295, Phe201, Ala203, Gln204, Thr207, His208, Phe211, Lys212, Thr213, Hie215, Tyr149, Leu409
|
7
|
− 11.284
|
− 71.663
|
Phe405, Phe396, Leu392, Leu391, Hie389, Trp388, Hie387, Tyr386, Tyr149, Asn383, Leu409, Ala200, Phe201, Ala203, Gln204, Thr207, His208, Phe211, Lys212, Thr213, Asp214, Hie215, Val296, Leu295, Val292, Glu291, Gln290, Ile275, Arg223, Val448
|
COH
|
− 8.93
|
− 54.81
|
Glu291, Lys216, Arg223, Lys212, Gln290, His 215
|
Raltitrexed (Tomudex)
|
− 10.83
|
− 58.73
|
Glu291, Arg223, Lys212, Gln290, Thr238, Glu 209
|
5-Fluorouracil
|
− 4.122
|
− 26.585
|
Leu392, Leu391, Hie389, Trp388, Hie387, Tyr386, Thr207, Gln204, Ala203, Ala200
|