Covalent inhibitors | Non covalent inhibitors | ||||
---|---|---|---|---|---|
Compound | Structure | References | Compound | Structure | References |
BTZ043 |
| [23] | 1–4 Azaindoles |
| [34] |
DNB1 |
| [35] | 2-Carboxyquinoxalines |
| [32] |
377790 |
| [26] | 4-AQs |
| [36] |
cBT |
| [16] | 8-Pyrrole-BTZ |
| [37] |
BTO |
| [38] | 1,3-BTZ azide |
| [39] |
VI-9376 |
| [40] | Pyrazolopyridones |
| [33] |
PBTZ |
| [17] | 1,2,4-Triazole containing 1,4-BTZ derivatives |
| [41] |