From: Therapeutic potential of heterocyclic pyrimidine scaffolds
Compound | IC50 (µmol/l) ± SD | |||
---|---|---|---|---|
H460 | HT-29 | MKN-45 | MDA-MB-231 | |
b31 | 0.057 ± 0.011 | 0.039 ± 0.008 | 0.25 ± 0.019 | 0.23 ± 0.020 |
GDC-0941 | 0.87 ± 0.20 | 0.86 ± 0.081 | 0.60 ± 0.12 | 0.28 ± 0.06 |
Sorafenib | 2.19 ± 0.11 | 3.61 ± 0.36 | 2.32 ± 0.35 | 0.94 ± 0.13 |