From: A new family of azanaphthoquinones for antimicrobial evaluation
Microorganisms | |||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|
Gram-negative bacteria | Gram-positive bacteria | Fungi | |||||||||
P. aeruginosa | E. coli | K. pneumoniae | P. mirabilis | S. aureus | S. epidermidis | E. faecalis | C. albicans | C. parapsilosis | C. tropicalis | ||
MIC values (μg/mL) | 3a | – | 156.2 | – | – | 156.2 | 2.44 | 39.06 | 78.12 | 78.12 | 39.06 |
3a′ | – | – | – | – | 312.5 | 156.2 | – | 312.5 | – | – | |
3b | – | 312.5 | – | – | 78.12 | 2.44 | 9.76 | 39.06 | 9.76 | 156.2 | |
3c | – | – | – | – | 39.06 | 39.06 | 156.2 | – | – | 312.5 | |
3d | – | – | – | – | 78.12 | 625 | 625 | – | – | – | |
3e | – | 156.2 | – | – | 312.5 | 39.06 | 312.5 | – | – | 312.5 | |
3e′ | – | – | – | – | 312.5 | 312.5 | – | – | – | 312.5 | |
3f | – | 312.5 | – | – | 312.5 | 1250 | 625 | – | 78.12 | – | |
3g | – | 156.2 | – | – | 312.5 | 19.53 | 625 | – | 156.2 | – | |
3h | – | – | 625 | – | 39.06 | 4.88 | 39.06 | – | 156.2 | 312.5 | |
3i | – | – | – | – | 312.5 | 312.5 | 625 | – | 78.12 | 312.5 | |
3j | – | 312.5 | 625 | – | 39.06 | 19.53 | 312.5 | – | 156.2 | 312.5 | |
Reference Antimicrobials | 2.4 Ceftazidime | 4.9 Cefuroxime-Na | 4.9 Cefuroxime-Na | 2.4 Cefuroxime-Na | 1.2 Cefuroxime-Na | 9.8 Cefuroxime | 128 Amikacin | 4.9 Clotrimazole | 0.5 Amphotericin B | 1 Amphotericin B |