Entry | No | Compound 5 | Yield (%) | Entry | No | Compound 6 | Yield (%) |
---|---|---|---|---|---|---|---|
1 | 5a |
| 74 | 12 | 6a |
| 50 |
2 | 5b |
| 95 | 13 | 6b |
| 30 |
3 | 5c |
| 95 | 14 | 6c |
| 29 |
4 | 5d |
| 90 | 15 | 6d |
| 28 |
5 | 5e |
| 87 | 16 | 6e |
| 33 |
6 | 5f |
| 91 | 17 | 6f |
| 37 |
7 | 5g |
| 94 | 18 | 6g |
| 50 |
8 | 5h |
| 93 | 19 | 6h |
| 50 |
9 | 5i |
| 93 | 20 | 6i |
| 6 |
10 | 5j |
| 79 | 21 | 6j |
| 54 |
11 | 5k |
| 89 | 22 | 6k |
| 52 |